at Peking University School of Pharmaceutical Sciences
the Jia Research Group
Independent research
104. “Design, syntheses and biological evaluation of natural product aiphanol derivatives and analogues: Discovery of potent anticancer agents”, Licheng Yao, Wenqing Cai, Shanmei Chen, Aidan Wang, Xin Wang, Chuanke Zhao, Chengchao Shou*, Yanxing Jia*. Bioorg. Med. Chem. Lett. 2023, 90, 129326.
103. “Total Synthesis of (+)-Aberrarone”, Yang Wang, Yongjian Su, Yanxing Jia*. J. Am. Chem. Soc. 2023, 145, 9459-9463.
102. “Total Synthesis of (−)-Principinol C”, Tianhao Ma , Hao Cheng , Mallesham Pitchakuntla , Weihao Ma , Yanxing Jia*. J. Am. Chem. Soc. 2022, 144, 20196-20200.
101. “Divergent Total Synthesis of Four Kopsane Alkaloids: N-Carbomethoxy-10,22-dioxokopsane, Epikopsanol-10-lactam, 10,22-Dioxokopsane, and N-Methylkopsanone”, Bo Qin, Zhepei Lu, Yanxing Jia*. Angew. Chem. Int. Ed. 2022, 61, e202201712.
100. “Bioinspired Total Synthesis of (+)-Euphorikanin A”, Zhuang Chen, Kuan Zhao, Yanxing Jia*. Angew. Chem. Int. Ed. 2022, 61, e202200576.
99. “Cascade Cyclization Reaction Initiated by Benzylic Carbocation of Indole: Scope and Mechanistic Insights”, Zhongrun Gao, Yuan Wang, Hang Song, Zhengren Xu*, Yanxing Jia*. Chin. J. Org. Chem. 2021, 41, 3126-3133.
98. “Protecting-Group-Free Total Synthesis of (–)-Pallambins A-D”, Xiwu Zhang, Yuan Wang, Peng Chen, Xinxian Cai, Yanxing Jia*. Chin. J. Chem. 2021, 39, 1983-1996.
97. “Total synthesis of Kopsine, Fruticosine, and structurally related polycyclic caged Kopsia indole alkaloids”, Bo Qin, Yuan Wang, Xin Wang*, Yanxing Jia*. Org. Chem. Front. 2021, 8(2), 369-383.
96. “Synthesis of benzofuro[3,2-b]indolines via regioselective electrooxidative coupling of indoles and phenols”, Keyuan Li, Yuan Wang, Lijun Chen, Lei Li, Yanxing Jia*. Tetrahedron. Lett. 2021, 63(36), 152603.
95. “Total Synthesis of (−)-Glaucocalyxin A”, Jiuzhou Guo, Bo Li, Weihao Ma, Mallesham Pitchakuntla, Yanxing Jia*. Angew. Chem. Int. Ed. 2020, 59(35), 15195–15198. Angew. Chem. 2020, 132(35), 15307–15310.
highlighted in synfacts, Synfacts 2020, 16(08), 0882.
《有机化学》亮点介绍，2020, 40(10), 3487-3489.
94. “Seven-step total synthesis of α-cyclopiazonic acid”, Shibin Shi, Kuo Yuan, Yanxing Jia*. Chin. Chem. Lett. 2020, 31(2), 401–403.
93. “A concise total synthesis of secoisolariciresinol”, Jiuzhou Guo, Yanxing Jia*. J. Chin. Pharm. Sci. 2019, 28(10), 699–703.
92. “Improved synthesis of key intermediate of grayanotoxin III”, Weihao Ma, Zhi Huang, Yanxing Jia*. J. Chin. Pharm. Sci. 2019, 28(6), 402–407.
91. “Type-II Pauson-Khand Reaction of 1,8-enyne in the Attempt of Building 7/5 Ring of (-)-Caribenol A and DFT Understanding”, Yang Wang, Kang Liu, Zhi-Xiang Yu*, Yanxing Jia*. Tetrahedron Lett. 2019, 60(36), 151001 .
90. “Natural product incarvillateine aggravates epileptic seizures by inhibiting GABAA currents”, Xiling Bian*, Yu Zhang, Bin Huang, Xintong Wang, Gongxin Wang, Yuhao Zhu, Yan Liu, Jianhui Liang, Yanxing Jia*, Kewei Wang*. Eur. J. Pharmaco. 2019, 858, 172496.
89. “Enantioselective Total Syntheses of Pallambins A-D”, Xiwu Zhang, Xinxian Cai, Bin Huang, Lei Guo, Zhongrun Gao, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(38), 13380–13384. Angew. Chem. 2019, 131(38), 13514–13518.
88. “A Ten-Step Total Synthesis of Speradine C”, Haichao Liu, Lijun Chen, Kuo Yuan, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(19), 6362–6365. Angew. Chem. 2019, 131(19), 6428–6431.
highlighted in synfacts, Synfacts 2019, 15(7), 0714.
《有机化学》亮点介绍，2019, 39(8), 2344.
87. “Eight-Step Total Synthesis of Phalarine by Bioinspired Oxidative Coupling of Indole and Phenol”, Lei Li, Kuo Yuan, Qianlan Jia, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(18), 6074–6078. Angew. Chem. 2019, 131(18), 6135–6139.
highlighted in synfacts, Synfacts 2019, 15(7), 0712.
x-mol化学资讯平台亮点介绍.
86. “Synthetic approaches to natural products containing a 2,3-dihydrobenzofuran skeleton”, Zhuang Chen, Mallesham Pitchakuntla, Yanxing Jia*. Nat. Prod. Rep. 2019, 36(4), 666–690.
85. “Recent Progress in the Synthesis of 3,4-Fused Indole Alkaloids” “3,4-桥环吲哚类生物碱的合成进展”, Kuo Yuan, Yanxing Jia*. Chin. J. Org. Chem. 2018, 38(9), 2386-2399. 《有机化学》，2018, 38(9), 2386-2399.
84. “Divergent Strategy in Natural Product Total Synthesis”, Lei Li, Zhuang Chen, Xiwu Zhang, Yanxing Jia*. Chem. Rev. 2018, 118(7), 3752–3832.
83. “Synthetic Study toward the Total Synthesis of Fumigaclavines A–D”, Yongfan Ma, Yanxing Jia*. J. Chin. Pharm. Sci. 2017, 26(7), 496–503.
82. “Regioselective Direct C-4 Functionalization of Indole: Total Syntheses of (–)-Agroclavine and (–)-Elymoclavine”, Jianbo Lv, Bin Wang, Kuo Yuan, Yuan Wang, Yanxing Jia*. Org. Lett. 2017, 19(13), 3664– 3667.
81.“Total Syntheses of Festuclavine, Pyroclavine, Costaclavine, epi-Costaclavine, Pibocin A, 9-Deacetoxyfumigaclavine C, Fumigaclavine G, and Dihydrosetoclavine”, Haichao Liu, Xiwu Zhang, Dong Shan, Mallesham Pitchakuntla, Yongfan Ma, Yanxing Jia*. Org. Lett. 2017, 19(12), 3323–3326.
80. “Total Syntheses of Naucleamides A−C and E, Geissoschizine, Geissoschizol, (E)-Isositsirikine, and 16-epi-(E)-Isositsirikine”, Lei Li, Paruke Aibibula, Qianlan Jia, Yanxing Jia*. Org. Lett. 2017, 19(10), 2642– 2645.
79.“Total synthesis of natural spiro-trisindole enantiomers similisines A, B and their stereoisomers”, Lunyong Shi, Lingyu Li, Jun Wang, Bin Huang, Kewu Zeng, Hongwei Jin, Qingying Zhang*, Yanxing Jia*. Tetrahedron Lett. 2017, 58(20), 1934–1938.
78. “Ergot alkaloids: synthetic approaches to lysergic acid and clavine alkaloids”, Haichao Liu, Yanxing Jia*. Nat. Prod. Rep. 2017, 34(4), 411–432.
77. “A Simple and Efficient Synthesis of Secondary Alkylamines from Nitroalkanes”, Zhi Huang, Jianbo Lu, Yanxing Jia*. ChemistrySelect. 2016, 1(18), 5892–5894.
76. “A concise gram-scale synthesis of ht-13-A via a rhodium-catalyzed intramolecular C–H activation reaction”, Pengyu Tao, Zhuang Chen, Yanxing Jia*. Chem. Commun. 2016, 52(75), 11300–11303.
75. “C–H bond activation in the total syntheses of natural products”, Pengyu Tao, Yanxing Jia*. Sci. China Chem. 2016, 59(9), 1109–1125.