at Peking University School of Pharmaceutical Sciences
中文版
​​​​the Jia Research Group
Independent research
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97. “Total synthesis of Kopsine, Fruticosine, and structurally related polycyclic caged Kopsia indole alkaloids”, Bo Qin, Yuan Wang, Xin Wang*, Yanxing Jia*. Org. Chem. Front. 2021, 8(2), 3​69-383.
96. “Synthesis of benzofuro[3,2-b]indolines via regioselective electrooxidative coupling of indoles and phenols”, Keyuan Li, Yuan Wang, Lijun Chen, Lei Li, Yanxing Jia*. Tetrahedron. Lett. 2021, 63(36), 152603.
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95. “Total Synthesis of (−)-Glaucocalyxin A”, Jiuzhou Guo, Bo Li, Weihao Ma, Mallesham Pitchakuntla, Yanxing Jia*. Angew. Chem. Int. Ed. 2020, 59(35), 15195–15198. Angew. Chem. 2020, 132(35), 15307–15310.

highlighted in synfacts, Synfacts 2020, 16(08), 0882.

《有机化学》亮点介绍2020, 40(10), 3487-3489.

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94. “Seven-step total synthesis of α-cyclopiazonic acid”, Shibin Shi, Kuo Yuan, Yanxing Jia*. Chin. Chem. Lett. 2020, 31(2), 401403.
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93. “A concise total synthesis of secoisolariciresinol”, Jiuzhou Guo, Yanxing Jia*. J. Chin. Pharm. Sci. 2019, 28(10), 699703.
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92. “Improved synthesis of key intermediate of grayanotoxin III”, Weihao Ma, Zhi Huang, Yanxing Jia*. J. Chin. Pharm. Sci. 2019, 28(6), 402407.
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91. “Type-II Pauson-Khand Reaction of 1,8-enyne in the Attempt of Building 7/5 Ring of (-)-Caribenol A and DFT Understanding”, Yang Wang, Kang Liu, Zhi-Xiang Yu*, Yanxing Jia*. Tetrahedron Lett. 2019, 60(36), 151001 .
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90. “Natural product incarvillateine aggravates epileptic seizures by inhibiting GABAA currents”, Xiling Bian*, Yu Zhang, Bin Huang, Xintong Wang, Gongxin Wang, Yuhao Zhu, Yan Liu, Jianhui Liang, Yanxing Jia*, Kewei Wang*. Eur. J. Pharmaco. 2019, 858, 172496.
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89. Enantioselective Total Syntheses of Pallambins A-D”, Xiwu Zhang, Xinxian Cai, Bin Huang, Lei Guo, Zhongrun Gao, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(38), 13380–13384. Angew. Chem. 2019, 131(38), 13514–13518.
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88. “A Ten-Step Total Synthesis of Speradine C”, Haichao Liu, Lijun Chen, Kuo Yuan, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(19), 6362–6365. Angew. Chem. 2019, 131(19), 6428–6431.

highlighted in synfacts, Synfacts 2019, 15(7), 0714.

     《有机化学》亮点介绍2019, 39(8), 2344.

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87. “Eight-Step Total Synthesis of Phalarine by Bioinspired Oxidative Coupling of Indole and Phenol”, Lei Li, Kuo Yuan, Qianlan Jia, Yanxing Jia*. Angew. Chem. Int. Ed. 2019, 58(18), 60746078. Angew. Chem. 2019, 131(18), 6135–6139.

highlighted in synfacts, Synfacts 2019, 15(7), 0712.

x-mol化学资讯平台亮点介绍.

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86. “Synthetic approaches to natural products containing a 2,3-dihydrobenzofuran skeleton”, Zhuang Chen, Mallesham Pitchakuntla, Yanxing Jia*. Nat. Prod. Rep. 2019, 36(4), 666690.
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85. “Recent Progress in the Synthesis of 3,4-Fused Indole Alkaloids 3,4-桥环吲哚类生物碱的合成进展, Kuo Yuan, Yanxing Jia*. Chin. J. Org. Chem. 2018, 38(9), 2386-2399. 《有机化学》,2018, 38(9), 2386-2399.
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84. “Divergent Strategy in Natural Product Total Synthesis”, Lei Li, Zhuang Chen, Xiwu Zhang, Yanxing Jia*. Chem. Rev. 2018, 118(7), 37523832.
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83. “Synthetic Study toward the Total Synthesis of Fumigaclavines A–D”, Yongfan Ma, Yanxing Jia*. J. Chin. Pharm. Sci. 2017, 26(7), 496503.
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82. “Regioselective Direct C-4 Functionalization of Indole: Total Syntheses of (–)-Agroclavine and (–)-Elymoclavine”, Jianbo Lv, Bin Wang, Kuo Yuan, Yuan Wang, Yanxing Jia*. Org. Lett. 2017, 19(13), 3664 3667.
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81.“Total Syntheses of Festuclavine, Pyroclavine, Costaclavine, epi-Costaclavine, Pibocin A, 9-Deacetoxyfumigaclavine C, Fumigaclavine G, and Dihydrosetoclavine”, Haichao Liu, X​​iwu Zhang, Dong Shan, Mallesham Pitchakuntla, Yongfan Ma, Yanxing Jia*. Org. Lett. 2017, 19(12), 33233326.
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80. “Total Syntheses of Naucleamides A−C and E, Geissoschizine, Geissoschizol, (E)-Isositsirikine, and 16-epi-(E)-Isositsirikine”, Lei Li, Paruke Aibibula, Qianlan Jia, Yanxing Jia*. Org. Lett. 2017, 19(10), 2642 2645.
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79.“Total synthesis of natural spiro-trisindole enantiomers similisines A, B and their stereoisomers”, Lunyong Shi, Lingyu Li, Jun Wang, Bin Huang, Kewu Zeng, Hongwei Jin, Qingying Zhang*, Yanxing Jia*. Tetrahedron Lett. 2017, 58(20), 1934–1938.
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78. “Ergot alkaloids: synthetic approaches to lysergic acid and clavine alkaloids, Haichao Liu, Yanxing Jia*. Nat. Prod. Rep. 2017, 34(4), 411432.
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77. “A Simple and Efficient Synthesis of Secondary Alkylamines from Nitroalkanes”, Zhi Huang, Jianbo Lu, Yanxing Jia*. ChemistrySelect. 2016, 1(18), 58925894.
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76. “A concise gram-scale synthesis of ht-13-A via a rhodium-catalyzed intramolecular CH activation reaction”, Pengyu Tao, Zhuang Chen, Yanxing Jia*. Chem. Commun. 2016, 52(75), 1130011303.
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75. “C–H bond activation in the total syntheses of natural products”, Pengyu Tao, Yanxing Jia*. Sci. China Chem. 2016, 59(9), 11091125.
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74. “A palladium-catalyzed intramolecular carbonylative annulation reaction to form 4,5-fused tricyclic 2-quinolones, Xiwu Zhang, Haichao Liu, Yanxing Jia*. Chem. Commun. 2016, 52(49), 76657667.

highlighted in synfacts, Synfacts 2016, 12(9), 0896.

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73. “Gram Scale Syntheses of (-)-Incarvillateine and Its Analogs. Discovery of Potent Analgesics for Neuropathic Pain”, Bin Huang, Fengying Zhang, Gang Yu, Yan Song, Xintong Wang, Meiliang Wang, Zehui Gong, Ruibin Su, Yanxing Jia*. J. Med. Chem. 2016, 59(8), 39533963 .
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72. “Asymmetric Total Synthesis of 3-epi-naucleamide A”, Paruke Aibibula, Zhi Huang, Hong-Zheng Fu,* Yanxing Jia*. J. Chin. Pharm. Sci. 2016, 25(1), 3036.
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71. “Formal Synthesis of (+)-Kopsihainanine A and Synthetic Study toward (+)-Limaspermidine”, Zhuang Chen, Shiqiang Zhou, Yanxing Jia*. J. Org. Chem. 2015, 80(24), 1254512551.
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70. “Antinociceptive effects of incarvillateine, a monoterpene alkaloid from Incarvillea sinensis, and possible involvement of the adenosine system”, Mei-Liang Wang, Gang Yu*, Shou-Pu Yi, Feng-Ying Zhang, Zhi-Tong Wang, Bin Huang, Rui-Bin Su*, Yan-Xing Jia, Ze-Hui Gong. Sci. Rep. 2015, 5, 16107.
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69.Protecting-Group-Free Enantioselective Synthesis of (-)-Pallavicinin and (+)-Neopallavicinin, Bin Huang, Lei Guo, Yanxing Jia*. Angew. Chem. Int. Ed. 2015, 54(46), 13599–13603. Angew. Chem. 2015, 127(46), 13803–13807.

(highlighted in synfacts, Synfacts 2015, 11(12), 1242.

Organic Chemistry Portal (http://www.organic-chemistry.org/Highlights /2016/01August. shtm), D. F. Taber,

x-mol化学资讯平台(http://www.x-mol.com/news/1398)亮点介绍 .

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68. “Catalytic Asymmetric Total Synthesis of (-)-Galanthamine and (-)-Lycoramine”, Lei Li, Qiao Yang, Yuan Wang, Yanxing Jia*. Angew. Chem. Int. Ed. 2015, 54(21), 62556259. Angew. Chem. 2015, 127(21), 6353–6357.

highlighted in synfacts, Synfacts 2015, 11(7), 0688.

Organic Chemistry Portalhttp://www.organic-chemistry.org/Highlights/2015 /30November.shtm

D. F. Taber, Org. Chem. Highlights 2015, November 30.